Lycorine Hydrochloride
Lycorine Hydrochloride ndeye chena kune-chena poda inobva kune alkaloid lycorine, iyo inowanikwa mune zvinomera zveLycris radiata radiata (l'her.), Uye ndezvemhuri yeAmarelliraeae. Lycorine Hydrochloride ine akasiyana mishonga yemishonga, kusanganisira anti-tumor, anti-cancer, anti-hutch, anti-buttus, anti-angiogensis, uye anti-marariya. Inonyura mumvura, Dmso, neEtazari. Chemakemikari chemuzvemakemikari chinoratidzwa neyakaomarara steroidal framework ine kuravira kwemapoka akawanda anoshanda, kusanganisira hydroxyl uye amino mapoka, zvichikonzera zviitiko zvayo zvezvisikwa.
Chigadzirwa Zita | Lycorine Hydrochloride Cas: 2188-68-3 | ||
STOURS SWOURSE | Lycris | ||
Kuchengetedza mamiriro | Chengetedza nechisimbiso pamhepo tembiricha | Chirevo Zuva | 2024.08.24 |
Chinhu | Standard | Mhedzisiro |
Kuchena(Hplc) | Lycorine Hydrochloride≥98% | 99,7% |
Chitarisiko | Off-chena poda | Kuwirirana |
Hunhu hwemuviriICS | ||
Chikamu-saizi | Nlt100% 80Mesh | Kuwirirana |
Kurasikirwa pakuoma | ≤1.0% | 1.8% |
Zvinorema simbi | ||
Yakazara simbi | ≤10.0PPMP | Kuwirirana |
Tungamira | ≤2.0PPMP | Kuwirirana |
Mercury | ≤1.0PPM | Kuwirirana |
Cadmium | ≤0.5PMP | Kuwirirana |
Microorganism | ||
Huwandu hwehutachiona hwehutachiona | ≤1000cfu / g | Kuwirirana |
Mbiriso | ≤100CFU / G | Kuwirirana |
Escherichia coli | Isina kubatanidzwa | Isina kuwonekwa |
Salmonella | Isina kubatanidzwa | Isina kuwonekwa |
Staphylococcus | Isina kubatanidzwa | Isina kuwonekwa |
Mhedziso | Vanokwanisa |
Zvimiro:
(1) kuchena kwakanyanya:Chigadzirwa chedu chinonyatsogadziriswa kuti uve nechokwadi chekuchena kwakanyanya, izvo zvakakosha pakubata kwayo uye kuchengeteka mumanyorero akasiyana siyana.
(2) anticancer zvivakwa:Izvo zvakaratidza kukosha kwehunyanzvi hwemhando dzakasiyana siyana dzemhando dzekenza, muVIVO uye muVivo, kuburikidza neVivo, kuburikidza nekusungwa kweCercle Clecle, kugadzirisa Aposis, uye inhibiting angiogenis.
(3) chiitiko chakaganhurika:Lycorine Hydrochloride inotendwa kuti ifambe neyakawandisa mamexcular tarisiro, ichipa chiitiko chevhu-spectrum inoshanda pamusoro pe cancer cancer cancer cancer cancer cancer.
(4) kuderera kwetsika:Izvo zvinoratidzira kudzikisira kwehupfumi kune zvakajairika masero, icho chinhu chakakosha pakushandisa kwayo seanoratidzira mumiriri.
(5) Pharmacokinetic profile:Chigadzirwa chacho chakadzidzwa kune yayo yemishonga yayo, kuratidza kukurumidza kutumira uye nekukurumidza kubviswa kubva plasma, izvo zvakakosha pakuronga uye kuronga kuronga.
(6) Mhedzisiro yeSynergistic:Lycorine Hydrochloride yakaratidza mamiriro akaisirwa kana achishandiswa pamwe chete nemimwe madhiragi, ayo anogona kubatsira mukukunda zvinodhaka uye kugadzirisa mabiko ekurapa.
(7) Tsvagurudzo-Yakatsigirwa:Chigadzirwa chinotsigirwa nekutsvagisa kwakawanda, kupa hwaro hwakasimba hwekushandiswa kwayo mukuvandudza mishonga uye clinical application.
(8) Ruzivo rwevimbiso:Rudzius mhando dzekudzora matanho ari munzvimbo mukati mekugadzirwa kwekugadzira kuti ive nechokwadi chekuenderana uye kuvimbika kwechigadzirwa.
(9) Zvikumbiro zvinokosha:Inokodzera kushandiswa mukutsvagisa nekuvandudza kwemibvunzo yekunyorera, kusanganisira kuwanikwa kwezvinodhaka uye kurapa kwekanza kurapwa.
(10) kutevedzera:Yakagadzirwa nekutevera gmp zviyero kuti uve nechokwadi chekuchengetedza kwechigadzirwa uye kushanda.
(1) Indasitiri yemishonga:Lycorine Hydrochloride inoshandiswa mukuvandudzwa kwemishonga yeAntiveral uye anticcancer mishonga.
(2) Biotechnology indasitiri:Iyo inoshandiswa mukutsvagisa uye kuvandudza kwevatsva vatsva vekurapa uye magadzirirwo ezvinodhaka.
(3) Chisiko chechigadzirwa chekutsvaga:Lycorine hydrochloride inodzidziswa nekuda kwehutano hwayo hutano uye mishonga yekurapa.
(4) Indasitiri yemakemikari:Inogona kushandiswa semakemikari epakati mune synthesis yemamwe makomendi.
(5) Indasitiri yekurima:Lycorine Hydrochloride yakafemerwa kuti igoneketi yayo sechipfuva chechisikigo uye chirimwa kukura kukura.
Iyo yekubvisa maitiro eLycorine Hydrochloride kazhinji inosanganisira inotevera nhanho nhanho kuti ive nekuchena kweiyo solvent uye kugadzirisa chiyero chekugadzirisa:
(1) Raw zvinyorwa zvekusarudza uye kunyepedzera:Sarudza yakakodzera Amarylliwaeaee chirimwa zvidzitiro, senge manhamba emitambo, uye geza, pakaoma uye uvapwanya kuti uve nekuchena kwezvinhu zvakadzvanywa uye nekuvhara hwaro hwekubvisa.
(2)Composite enzyme kunamatwa:Shandisa kuomesa enzymes (senge cellulase uye perctinase) kunyepedzera kuraswa zvishandiso zvekushongedza zvirimwa masero uye kugadzirisa zvinotevera zvibodzwa zvekushandisa.
(3)Dilute Hydrochloric Acid kusimuka:Sanganisa iyo yekunyepedzera yakasviba zvinhu ne dilute hydrochloric acid mhinduro yekubvisa lycorine. Iko kushandiswa kwehydrochloric acid kunobatsira kuwedzera iyo solubility ye lycorine, nokudaro ichivandudza kudzvanywa kwekunyatsojeka.
(4)Ultrasonic-yakabatsira kubviswa:Iko kushandiswa kweiyo ultrasonic tekinoroji yekuwedzera inogona kukurudzira maitiro ekunyungudza kwe lycorine mune solvent uye kugadzirisa kunyatsoita uye kuchena.
(5)Chloroform yekubvisa:Kuongororwa kunoitwa ne organic sol sol sol solorform, uye iyo lycorine inotamiswa kubva muchikamu chemaziso kune iyo organic chikamu kuti uwedzere kunatsa chinangwa.
(6)Solvent kupora:Mushure mekutora maitiro, iyo solvent yakadzoserwa kuburikidza nekuvapurwa kana distillation kuti uderedze solvent kushandiswa uye kugadzirisa hupfumi.
(7)Kucheneswa uye kuoma:Kuburikidza nekucheneswa kwakakodzera uye kuoma matanho, yakachena lycorine hydrochloride poda inowanikwa.
Mumamiriro ese ese ekutsanangurwa Iko kushandiswa kwezvino -zvazvino kubviswa uye nekuchenesa michina, sekuti seyakawedzera urefu
Chengetedza: Ramba uine inotonhorera, yakaoma, yakaoma nzvimbo nzvimbo, chengetedza kubva mukunyorova uye zvakananga mwenje.
Bulk package: 25kg / chigubhu.
Tungamira nguva: Mazuva manomwe mushure mekuraira kwako.
HEREF Hupenyu: makore maviri.
Remark: yakatarwa yakatarwa zvakare inogona kuwanikwa.

Taura
Pasi pe100kg, 3-5days
Gonhi rekushanda pasuo riri nyore kutora zvinhu
Negungwa
Over300kg, makore makumi matatu apfuura
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Nemhepo
100kg-1000kg, 5-7days
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Lycorine chiitiko chomuzvarirwo chinoitika alkaloid iyo inogona kuwanikwa mune dzinoverengeka zvidyarwa, kunyanya mukati memhuri yeAmarelloaceae. Hezvino zvimwe zvinomera zvinozivikanwa kuti zvine lycorine:
Lycris radiata.
Leucojum Aestivum(zhizha snowflake), rinozivikanwa kuti riine lycorine.
Ungernia sewarzowiiImwe chirimwa kubva kumhuri yeAmarellIdaae iyo yakataurwa kuti iite Lycorine.
Hippeastrum hybrid (iyo Isita Lily)Uye zvimwe zvinongedzo zvine chekuita nezvirimwa zvinozivikanwa zvitsva zve lycorine.
Izvi zvirimwa zvinogoverwa zvakanyanya munzvimbo dzinopisa uye dzakazara pasi rese uye dzive nenhoroondo refu yekushandiswa mumushonga wetsika. Kuvapo kweRycorine mune izvi zvidyarwa kwave kuri nyaya yekutsvagisa nekuda kwezvakangoita zve pharmacological zvivakwa, kusanganisira yakakosha anticancer mhedzisiro sezvakaratidzwa muzvidzidzo zvakasiyana.
Lycorine ndeyechisikigo alkaloid ine huwandu hwakawanda hwemagetsi, kusanganisira zvayo zvinogona kushandiswa mu cancer kurapwa. Nechinoratidza kuvimbisa zvinoguma nekudzidza kwakasiyana siyana, kune mamwe mimwe mhedzisiro uye kufunga kwakabatana nekushandiswa kwayo:
Kuderera Kwemhando: Lycorine uye yayo Hydrochloride Munyu unowanzo kuratidzira kuderera kwehupfumi, iyo iri hunhu hwakanaka hwekushandisa kiriniki. Izvo zvakaratidzirwa kuve nemhedzisiro midiki pane zvakajairwa masero emunhu uye makonzo ane hutano, achiratidza rimwe danho rekusarudzika kwemasero ematehwe pamusoro peyakajairwa.
NYAYA YEMADZIMAI YEMAHARA
Hapana hurongwa hwemotokari kusanzwisisika: zvidzidzo zvakaratidza kuti serial doses of lycorine hazvikanganwe kusanzwisisika kwemotokari, zvichiratidza kuti hazvitungamire kuCentraus system (CNS) mhedzisiro inoenderana nemotokari kudzora kwemotokari.
Chinoita kuti ubatanidzane
Kuzvibata kwakajairika uye kunyatsoita
Hapana akakosha akakosha pamari yehuremu kana hutano hweLycorine uye Lycorine Hydrochloride haana kukonzeresa huremu kana huwandu hwehutano hwemuviri mune bundu rombo.
Izvo zvakakosha kuti uzive kuti nepo lycorine yakaratidza mukana mukuongorora kwepamberi, ongororo kwenguva refu yekuongorora ichiri kuderera. Kuwedzera kutsvagisa kunodiwa kunyatsonzwisisa chimiro chayo chekuchengetedza, kunyanya kushandiswa kwenguva refu uye mumakiriniki marongero. Mhedzisiro uye kuchengetedzwa kwe lycorine kunogona kusiyana zvichienderana neshiri, nzira yekutonga, uye hunhu hwemurwere. Gara uchibvunza neine hutano hwehutano hwekufunga usati wafunga nezvekushandiswa kwe chero chitsva chekuwedzera kana kurapwa.